Synthesis of 5-(pyrazol-1-yl)-1,2,3-thiadiazoles / Vysokova Olga A.,Kalinina Tatiana A.,Tokareva Marina A.,Pospelova Tatiana A.,Glukhareva Tatiana V.,Morzherin Yuri Yu. // CHEMISTRY OF HETEROCYCLIC COMPOUNDS. - 2017. - V. 53, l. 2. - P. 236-238.

ISSN/EISSN:

0009-3122 / 1573-8353

Type:

Article

Abstract:

method is proposed for the synthesis of ethyl 5-(3-aryl-4-formyl-1H-pyrazol-1- yl)-1,2,3-thiadiazole-4-carboxylates by a reaction of acetophenone (4-ethoxycarbonyl-1,2,3-thiadiazol-5-yl)hydrazones with a Vilsmeier-Haack complex. The obtained heterocyclic assemblies provide interesting substrates for further modification and study of biological activity.

Author keywords:

heterocyclic assemblies; acetophenone hydrazones; 5-(pyrazol-1-yl)-1,2,3-thiadiazoles; pyrazoles; 1,2,3-thiadiazoles; Vilsmeier-Haack reaction DERIVATIVES; 1,2,3-THIADIAZOLE; BIOACTIVITIES; INHIBITORS; MOIETY

DOI:

10.1007/s10593-017-2045-5

Web of Science ID:

ISI:000397339800018

Соавторы в МНС:

Другие поля

Поле	Значение
Month	FEB
Publisher	SPRINGER
Address	233 SPRING ST, NEW YORK, NY 10013 USA
Language	English
EISSN	1573-8353
Keywords-Plus	DERIVATIVES; 1,2,3-THIADIAZOLE; BIOACTIVITIES; INHIBITORS; MOIETY
Research-Areas	Chemistry
Web-of-Science-Categories	Chemistry, Organic
Author-Email	taniagluhareva@yandex.ru
Funding-Acknowledgement	Russian Science Foundation {[}16-16-04022]
Funding-Text	This work was performed with financial support from the Russian Science Foundation (grant 16-16-04022).
Number-of-Cited-References	12
Usage-Count-Last-180-days	1
Usage-Count-Since-2013	1
Journal-ISO	Chem. Heterocycl. Compds.
Doc-Delivery-Number	EP4GU