Synthesis of 5-(pyrazol-1-yl)-1,2,3-thiadiazoles / Vysokova O.A., Kalinina T.A., Tokareva M.A., Pospelova T.A., Glukhareva T.V., Morzherin Y.Y. // Chemistry of Heterocyclic Compounds. - 2017. - V. 53, l. 2. - P. 236-238.

ISSN:

00093122

Type:

Article

Abstract:

[Figure not available: see fulltext.] A method is proposed for the synthesis of ethyl 5-(3-aryl-4-formyl-1H-pyrazol-1-yl)-1,2,3-thiadiazole-4-carboxylates by a reaction of acetophenone (4-ethoxycarbonyl-1,2,3-thiadiazol-5-yl)hydrazones with a Vilsmeier–Haack complex. The obtained heterocyclic assemblies provide interesting substrates for further modification and study of biological activity. © 2017, Springer Science+Business Media New York.

Author keywords:

1,2,3-thiadiazoles; 5-(pyrazol-1-yl)-1,2,3-thiadiazoles; acetophenone hydrazones; heterocyclic assemblies; pyrazoles; Vilsmeier–Haack reaction

Index keywords:

нет данных

DOI:

10.1007/s10593-017-2045-5

Смотреть в Scopus:

https://www.scopus.com/inward/record.uri?eid=2-s2.0-85015667902&doi=10.1007%2fs10593-017-2045-5&partnerID=40&md5=1b5384554b0460697e8f12495da7736d

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Link	https://www.scopus.com/inward/record.uri?eid=2-s2.0-85015667902&doi=10.1007%2fs10593-017-2045-5&partnerID=40&md5=1b5384554b0460697e8f12495da7736d
Affiliations	Ural Federal University named after the First President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg, Russian Federation
Author Keywords	1,2,3-thiadiazoles; 5-(pyrazol-1-yl)-1,2,3-thiadiazoles; acetophenone hydrazones; heterocyclic assemblies; pyrazoles; Vilsmeier–Haack reaction
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Correspondence Address	Glukhareva, T.V.; Ural Federal University named after the First President of Russia B. N. Yeltsin, 19 Mira St., Russian Federation; email: taniagluhareva@yandex.ru
Publisher	Springer New York LLC
CODEN	CHCCA
Language of Original Document	English
Abbreviated Source Title	Chem. Heterocycl. Compd.
Source	Scopus