Regioselective synthesis of trifluoromethylated 3-(pyrazolyl)indoles on the basis of 6-(trifluoromethyl)comanic acid / Usachev Boris I.,Obydennov Dmitrii L.,Sosnovskikh Vyacheslav Ya. // JOURNAL OF FLUORINE CHEMISTRY. - 2012. - V. 135, l. . - P. 278-284.

ISSN/EISSN:

0022-1139 / нет данных

Type:

Article

Abstract:

A number of trifluoromethylated 3-(pyrazolyl)indoles was synthesized from 2-(trifluoromethyl)comanic acid, its ethyl ester and amide via intermediate isomeric 5(3)-{[}3,3,3-trifluoro-2-(phenylhydrazono)-propyl]pyrazole-3(5)-carboxy lic acids and their derivatives. (C) 2011 Elsevier B.V. All rights reserved.

Author keywords:

6-(Trifluoromethyl)comanic acid; 3-(Pyrazolyl)indoles; Trifluoromethylated heterocycles; Fischer reaction; Regioselectivity PALLADIUM-CATALYZED ANNULATION; INDOLE-DERIVATIVES; AROMATIC-COMPOUNDS; INTERNAL ALKYNES; HETEROCYCLES; ENAMINES; ANTIFUNGAL

DOI:

10.1016/j.jfluchem.2011.12.008

Web of Science ID:

ISI:000301806400038

Соавторы в МНС:

Другие поля

Поле	Значение
Month	MAR
Publisher	ELSEVIER SCIENCE SA
Address	PO BOX 564, 1001 LAUSANNE, SWITZERLAND
Language	English
Keywords-Plus	PALLADIUM-CATALYZED ANNULATION; INDOLE-DERIVATIVES; AROMATIC-COMPOUNDS; INTERNAL ALKYNES; HETEROCYCLES; ENAMINES; ANTIFUNGAL
Research-Areas	Chemistry
Web-of-Science-Categories	Chemistry, Inorganic \& Nuclear; Chemistry, Organic
Author-Email	boris.usachev@mail.ru
Funding-Acknowledgement	Ministry of Education and Science {[}Pi1370]
Funding-Text	This work was financially supported by the Ministry of Education and Science (Contract No. Pi 1370).
Number-of-Cited-References	43
Usage-Count-Since-2013	5
Journal-ISO	J. Fluor. Chem.
Doc-Delivery-Number	912NH