Synthesis of 6-thienyl-substituted 2-amino-3-cyanopyridines / Verbitskiy E. V.,Cheprakova E. M.,Pervova M. G.,Danagulyan G. G.,Rusinov G. L.,Chupakhin O. N.,Charushin V. N. // RUSSIAN CHEMICAL BULLETIN. - 2015. - V. 64, l. 3. - P. 689-694.

ISSN/EISSN:
1066-5285 / 1573-9171
Type:
Article
Abstract:
An efficient method for the synthesis of 6-thienyl-substituted 2-amino-3-cyanopyridines by the ring transformation in the corresponding pyrimidines was developed. Further modification of the pyridines obtained under conditions of a room temperature aerobic Suzuki reaction in the presence of trans-bis(dicyclohexylamine) palladium(II) acetate as a catalyst was studied.
Author keywords:
pyrimidines; pyridines; transformations of heterocycle; Suzuki cross-coupling; trans-bis(dicyclohexylamine)palladium(II) acetate PYRIDINE-DERIVATIVES; RING TRANSFORMATIONS; 2-AMINONICOTINONITRILES; 5-NITROPYRIMIDINE
DOI:
10.1007/s11172-015-0920-8
Web of Science ID:
ISI:000365184100029
Соавторы в МНС:
Другие поля
Поле Значение
Month MAR
Publisher SPRINGER
Address 233 SPRING ST, NEW YORK, NY 10013 USA
Language English
EISSN 1573-9171
Keywords-Plus PYRIDINE-DERIVATIVES; RING TRANSFORMATIONS; 2-AMINONICOTINONITRILES; 5-NITROPYRIMIDINE
Research-Areas Chemistry
Web-of-Science-Categories Chemistry, Multidisciplinary
Author-Email Verbitsky@ios.uran.ru
Funding-Acknowledgement Ural Branch of the Russian Academy of Sciences {[}13-3-019-UMA]; Russian Foundation for Basic Research {[}13-03-96049-r\_ural\_a, 13-03-90606-Arm\_a, 14-03-31040-mol\_a]; Russian Federation {[}MK-3939.2014.3]; Skolkovo Institute of Science and Technologies; M. V. Lomonosov Moscow State University {[}182-MRA]
Funding-Text This work was financially supported by the Ural Branch of the Russian Academy of Sciences (Program 13-3-019-UMA), the Russian Foundation for Basic Research (Project Nos 13-03-96049-r\_ural\_a, 13-03-90606-Arm\_a, and 14-03-31040-mol\_a), the President of the Russian Federation Council for Grants (Program of State Support for Young Scientists-Candidates of Science, Grant MK-3939.2014.3), as well as within the Agreement between the Skolkovo Institute of Science and Technologies and the M. V. Lomonosov Moscow State University (No. 182-MRA).
Number-of-Cited-References 20
Usage-Count-Last-180-days 1
Usage-Count-Since-2013 4
Journal-ISO Russ. Chem. Bull.
Doc-Delivery-Number CW7MU